Biomedicinal Chemistry (Theory)

Drugs Acting on the Central Nervous System General Anesthetics Halothane, Methoxyflurane, Enflurane, Sevoflurane, Isoflurane, Desflurane, Methohexital, Thiamylal, Thiopental, Ketamine*, Ramelteon, Remimazolam, Fospropofol, Dexmedetomidine Sedatives and Hypnotics Barbital, Phenobarbital*, Mephobarbital, Amobarbital, Butabarbital, Pentobarbital, Secobarbital, Chlordiazepoxide, Diazepam*, Oxazepam, Chlorazepate, Lorazepam, Alprazolam, Zolpidem, Glutethimide, Meprobamate, Ethchlorvynol, Triclofos, Paraldehyde SAR of Barbiturates and Benzodiazepines Antipsychotics Promazine, Chlorpromazine*, Triflupromazine, Thioridazine, Piperacetazine, Prochlorperazine, Trifluoperazine, Chlorprothixene, Thiothixene, Loxapine, Clozapine, Haloperidol, Droperidol, Risperidone, Molindone, Sulpiride, Brexpiprazole, Lumateperone, Pimavanserin, Samidorphan SAR of Phenothiazines Anticonvulsants Phenobarbitone, Methabarbital, Phenytoin*, Mephenytoin, Ethotoin, Oxazolidinediones: Trimethadione, Paramethadione Succinimides: Phensuximide, Methsuximide, Ethosuximide Phenacemide, Carbamazepine*, Clonazepam, Primidone, Valproic acid, Gabapentin, Felbamate, Perampanel, Lacosamide, Retigabine SAR of Anticonvulsants

Anti-Infective Chemotherapeutic Agents Antitubercular Agents Isoniazid*, Ethionamide, Ethambutol, Pyrazinamide, Para-amino salicylic acid*, Rifampicin, Rifabutin, Cycloserine, Streptomycin, Capreomycin, Pretomanid, Clofazimine, Levofloxacin, Bedaquiline, Linezolid, Delamanid Antimalarials Quinine, Chloroquine*, Amodiaquine, Primaquine, Pamaquine, Quinacrine, Mefloquine, Cycloguanil pamoate, Proguanil, Pyrimethamine, Artesunate, Artemether, Atovaquone SAR of Quinoline derivatives Antiprotozoals Metronidazole*, Tinidazole, Ornidazole, Diloxanide, Iodoquinol, Pentamidine isethionate, Atovaquone,Eflornithine, Paromomycin, Nitazoxanide Antivirals Amantadine, Rimantadine, Idoxuridine, Acyclovir*, Ganciclovir, Zidovudine, Didanosine, Zalcitabine, Lamivudine,Loviride, Delavirdine, Ribavirin, Saquinavir, Indinavir, Ritonavir, Valganciclovir, Peramivir, Lenacapavir Antifungals Amphotericin-B, Nystatin, Natamycin, Griseofulvin, Clotrimazole, Econazole, Butoconazole, Oxiconazole, Tioconazole, Miconazole, Ketoconazole*, Terconazole, Itraconazole, Fluconazole, Naftifine, Tolnaftate, Posaconazole, Isavuconazole Anthelmintics Diethylcarbamazine, Thiabendazole, Mebendazole, Albendazole*, Niclosamide, Oxamniquine, Praziquantel, Ivermectin Urinary Tract Anti-infective Agents Nalidixic acid, Norfloxacin, Enoxacin, Ciprofloxacin*, Ofloxacin, Lomefloxacin, Sparfloxacin, Gatifloxacin, Furazolidone, Nitrofurantoin, Methenamine, Moxifloxacin SAR of Quinolones

Antibiotics and Sulfa Drugs Antibiotics -Lactamase inhibitors, Monobactams Aminoglycosides: Streptomycin, Neomycin, Kanamycin, Tetracyclines: Tetracycline, Oxytetracycline, Minocycline, Doxycycline, Macrolides: Erythromycin, Clarithromycin, Azithromycin Chloramphenicol*, Clindamycin, Clavulanic acid SAR of Penicillins, Tetracyclines, and Cephalosporins Sulfa Drugs Sulphamethizole, Sulfisoxazole, Sulphapyridine, Sulphathiazole, Sulfacetamide, Sulphamethoxazole,Sulphadiazine, Mefenide, Sulfasalazine, Trimethoprim, Cotrimoxazole, Dapsone* SAR of Sulfonamides

Antineoplastic Agents Mechlorethamine, Cyclophosphamide, Melphalan, Chlorambucil, Busulfan, Thiotepa, Mercaptopurine*, Thioguanine, Fluorouracil, Floxuridine, Cytarabine, Methotrexate*, Azathioprine, Dactinomycin, Daunorubicin, Doxorubicin, Bleomycin, Etoposide, Vinblastine, Vincristine, Paclitaxel, Camptothecin, Cisplatin, Mitotane, Carboplatin

Endocrine Drugs, Antidiabetic Agents and Narcotic Analgesics Endocrine Drugs Sex hormones: Testosterone, Nandrolone, Progesterone, Oestriol, Oestradiol, Oestrone, Diethylstilbestrol Drugs for erectile dysfunction: Sildenafil, Tadalafil Oral contraceptives: Mifepristone, Norgestrel, Levonorgestrel Corticosteroids: Cortisone, Hydrocortisone, Prednisolone, Betamethasone, Dexamethasone Thyroid and antithyroid drugs: L-Thyroxine, L-Thyronine, Propylthiouracil, Methimazole Antidiabetic Agents Insulin and preparations, Tolbutamide*, Chlorpropamide, Glipizide, Glimepiride Biguanides: Metformin Thiazolidinediones: Pioglitazone, Rosiglitazone Repaglinide, Nateglinide, Acarbose, Voglibose Narcotic Analgesics Morphine, Codeine, Meperidine, Anilerdine, Diphenoxylate, Loperamide, Fentanyl*, Methadone, Propoxyphene, Pentazocine, Levorphanol Nalorphine, Levallorphan, Naloxone SAR of Morphine analogues